Ligand efficiency as a guide in fragment hit selection and optimization.
نویسندگان
چکیده
Ligand efficiency as a guide in fragment hit selection and optimization Sabine Schultes, Chris de Graaf, Eric E.J. Haaksma*, Iwan J.P. de Esch, Rob Leurs, Oliver Krämer Boehringer Ingelheim RCV GmbH & Co. KG, Department of Medicinal Chemistry, Dr. Boehringer-Gasse 5-11, Vienna, Austria Leiden/Amsterdam Center for Drug Research (LACDR), Division of Medicinal Chemistry, Department of Pharmacochemistry, Faculty of Exact Sciences, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands Drug Discovery Today: Technologies Vol. 7, No. 3 2010
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ورودعنوان ژورنال:
- Drug discovery today. Technologies
دوره 7 3 شماره
صفحات -
تاریخ انتشار 2010